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Mononuclear rearrangement of heterocycles in zwitterionic micelles of amine oxide surfactants

Year: 2012

Journal: Journal of Colloid and Interface Science 2012, 381 (1) pp 67-72, 20121211

Authors: Susanna Guernelli, Antonella Fontana, Renato Noto, Domenico Spinelli, Maria Liria Turco Liveri

Organizations: Dipartimento di Chimica Organica “A. Mangini”, Università degli Studi di Bologna, Via S. Giacomo 11, 40126 Bologna, Italy, Dipartimento di Scienze del Farmaco, Università “G. d’Annunzio”, Via dei Vestini 31, 66013 Chieti, Italy, Dipartimento di Scienze e Tecnologie Molecolari e Biomolecolari (STEMBIO), Viale delle Scienze, Ed. 16, Parco d’Orleans 2, 90128 Palermo, Italy, Dipartimento di Chimica “G. Ciamician”, Università degli Studi di Bologna, Via Selmi 2, 40126 Bologna, Italy, Dipartimento di Chimica “S. Cannizzaro”, Viale delle Scienze, Ed. 17, Parco d’Orleans 2, 90128 Palermo, Italy

Rate constants for the mononuclearrearrangement (MRH) of Z-phenylhydrazones of some 5-substituted-3-benzoyl-1,2,4-oxadiazoles in water have been measured in the presence of zwitterionicmicelles. The use of micellized N-tetradecyl-N,N-dimethylamineoxide (C14DMAO) as the reaction medium allowed to solubilize the otherwise water-insoluble oxadiazoles. Micellar rate effects were analyzed by using a simple pseudo-phase model and compared with those obtained in non-ionic micelles (Triton X-100). Evidence that both the rate of the rearrangement reaction and the binding of the substrates to the micelles are mainly governed by substrate hydrophobicity is obtained. The disagreement with the primarily sterically controlled MRH in Triton X-100 micelles highlights large and intriguing differences between the two micellar environments.